Pharmacokinetics

Absorption: Well absorbed following oral administration. Food enhances absorption

Distribution: Unknown

Protein Binding: 99.9%

Metabolism and Excretion: Mostly metabolized by the liver (CYP3A4, CYP2C9 and CYP2C19 enzyme systems); minimal renal excretion; mostly eliminated in feces as unchanged drug and metabolites

Half-life: 41 hr

TIME/ACTION PROFILE (blood levels)

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